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2020


Maniindole, an indole derivative from the roots of Anonidium manii and combined antischistosomal and enzymatic activities
Josette Linda Toussi Matchi, Diderot Tchamo Noungoue, Isabelle Kuhn Jérôme Boissier, Jean Claude Tchouankeu, Marc Nothisen, Guilhem Chaubet, Delphine Garnier, Sylvain Ursuegui, Silvère Augustin, Alain Wagner; Nat. Prod. Res. 2020. 1-9.
Doi: 10.1080/14786419.2020.1824227

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Dual Gene Delivery Reagents From Antiproliferative Alkylphospholipids for Combined Antitumor Therapy
Boris Gaillard, Jean-Serge Remy, Françoise Pons, Luc Lebeau; Front. Chem. 2020. 8, 581260.
Doi: 10.3389/fchem.2020.581260


Synthesis and Evaluation of Antitumor Alkylphospholipid Prodrugs
Boris Gaillard, Jean-Serge Remy, Françoise Pons, Luc Lebeau; Pharm. Res. 2020. 37, 6, 106.
Doi.org/10.1007/s11095-020-02830-y


Investigating Ugi / Passerini multicomponent reactions for the Site‐Selective Conjugation of Native Trastuzumab
Charlotte Sornay, Steve Hessmann, Stéphane Erb, Igor Dovgan, Anthony Ehkirch, Thomas Botzanowski, Sarah Cianférani, Alain Wagner, Guilhem Chaubet; Chem. Eur. J. 2020. 26, 61, 13797-13805.
Doi:10.1002/chem.202002432

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On the use of DNA as a linker in antibody-drug conjugates: synthesis, stability and in vitro potency
Igor Dovgan, Anthony Ehkirch, Victor Lehot, Isabelle Kuhn, Oleksandr Koniev, Sergii Kolodych, Alexandre Hentz, Manon Ripoll, Sylvain Ursuegui, Marc Nothisen, Sarah Cianférani, Alain Wagner; Sci. Rep., 2020, 10, 7691.
Doi.org/10.1038/s41598-020-64518-y

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Ethynylation of Cysteine Residues: From Peptides to Proteins in Vitro and in Living Cells
Romain Tessier, Raj Kumar Nandi, Brendan G. Dwyer, Daniel Abegg, Charlotte Sornay, Javier Ceballos, Stephane Erb, Sarah Cianferani, Alain Wagner, Guilhem Chaubet, Alexander Adibekian, Jerome Waser; Angew. Chem. Int. Ed. 2020 , 59 , 10961.
Doi.org/10.1002/anie.202002626

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Automated linkage of proteins and payloads producing monodisperse conjugates
Igor Dovgan, Alexandre Hentz, Oleksandr Koniev, Anthony Ehkirch, Steve Hessmann, Sylvain Ursuegui, Sébastien Delacroix, Margaux Riomet, Frédéric Taran, Sarah Cianférani, Sergii Kolodych, Alain Wagner; Chem. Sci., 2020, 11, 1210-1215.
Doi: 10.1039/C9SC05468E

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2019


Antibody-Oligonucleotide Conjugates as Therapeutic, Imaging, and Detection Agents
Igor Dovgan, Oleksandr Koniev, Sergii Kolodych, Alain Wagner; Bioconjugate Chem., 2019, 30, 10, 2483-2501.
DOI: 10.1021/acs.bioconjchem.9b00306


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Design and evaluation of ionizable peptide amphiphiles for siRNA delivery.
Patrick Neuberg, Alain Wagner, Jean-Serge Remy, Antoine Kichler; Int. J. Pharmaceut., 2019, 566, 141-148.
DOI: 10.1016/j.ijpharm.2019.05.052
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​​Sydnone-based turn-on fluorogenic probes for no-wash protein labeling and in-cell imaging.
Lucie Plougastel, Manas R. Pattanayak, Margaux Riomet, Sarah Bregant, Antoine Sallustrau, Marc Nothisen, Alain Wagner, Davide Audisio, Frédéric Taran; Chem. Commun., 2018, 55, 4582-4585.
DOI:  10.1039/C9CC01458F

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2018


​​Synthesis and Kinetic evaluation of an azido analogue of methylerythritol phosphate: a Novel Inhibitor of E-coli YgbP/IspD
Zoljargal Baatarkhuu, Philippe Chaignon, Franck Borel, Jean-Luc Ferrer, Alain Wagner, Myriam Seemann; Scientific Reports, 2018, 8, 17892-17901.
DOI: 
10.1038/s41598-018-35586-y
038/s41598-018-35586-y  :10.1038/s41598-018-35586-y
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​​Co-delivery of anti-PLK-1 si RNA and camptothecin by nanometric polydiacetylenic micelles results in a synergistic cell killing
Manon Ripoll, Marie Pierdant, Patrick Neuberg, Dominique Bagnard, Alain Wagner, Antoine Kichler, Jean-Serge Remy; RSC Advances, 2018, 8, 20758-20763. 
DOI: 
 10.1039/c8ra03375g

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Expedient synthesis of trifunctional oligoethyleneglycol-amine linkers and their use in the preparation of PEG-based branched platforms
Sylvain Ursuegui, Jérémy P. Schneider, Claire Imbs, Florian Lauvoisard, Marta Dudek, Michel Mosser, Alain Wagner; Organic and Biomolecular Chemistry, 2018, 16, 8579-8584.
DOI: 
 10.1039/c8ob02097c

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Recent, non-classical, approaches to antibody lysine modification
Guilhem Chaubet, Fabien Thoreau, Alain Wagner; Drug Discovery Today: Technologies, 2018, 30, 21-26.
DOI: 10.1016/j.ddtec.2018.09.002
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Reduction Inhibition of dengue virus infection by mannoside glycolipid conjugates
Evelyne Schaeffer, Vincent Flacher, Patrick Neuberg, Astrid Hoste, Adrien Brulefert, Jean-Daniel Fauny, Alain Wagner, Christopher G. Mueller; Antiviral Research, 2018, 154, 116-123.
DOI: 10.1016/j.antiviral.2018.04.005


Reduction–rebridging strategy for the preparation of ADPN-based antibody–drug conjugates
Oleksandr Koniev, Igor Dovgan, Brigitte Renoux, Anthony Ehkirch, Jitka Eberova, Sarah Cianférani, Sergii Kolodych, Sébastien Papot and  Alain Wagner, Med. Chem. Commun., 2018, 9, 5, 827-830.
DOI:
10.1039/C8MD00141C
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Arginine-Selective Bioconjugation with 4-Azidophenyl glyoxal: Application to the single and Dual Functionalisation of Native Antibody
Igor Dovgan, Stéphane Erb, Steve Hessman, Sylvain Ursuegui, Chloé Michel, Christian Muller, Guilhem Chaubet, Sarah Cianférani and Alain Wagner, Organic & Biomolecular Chemistry, 2018, 16, 8, 1305-1311.
DOI: 10.1039/C7OB02844J

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Polydiacetylenic Nanofibers as New siRNA Vehicles for in vitro and  in vivo Delivery
E P. Neuberg, I. Hamaidi, D. Danilin, M. Ripoll, V. Lindner, M. Nothisen, A. Wagner, A. Kichler, T. Massfelder and J.-D. Remy, Nanoscale, 2018, 10, 1587-1590.
DOI: 
10.1039/C7NR09202D
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2017


Structural Investigation of Cyclo-dioxo Maleimide Cross-linkers for Acid and Serum Stability
Elisabetta Tobaldi, Igor Dovgan, Michel Mosser, Jean-Michel Becht, Alain Wagner, Organic & Biomolecular Chemistry, 2017, 15, 9305-9310.
DOI: 10.1039/c7ob01757j
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Discovery of New Click and Release Reactions by Screening of Mesoionics and Cycloalkynes Combinations 
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Frédéric Taran, Sabrina Bernard, Davide Audisio, Riomet Margaux, Sarah Bregant, Antoine Sallustrau, Lucie Plougastel, Elodie Decuypere, Sandra Gabillet, Ramar Arun Kumar, Jijy Elyian, Minh Nguyet Trinh, Oleksandr Koniev, Alain Wagner, Sergii Kolodych,
Angewandte Chemie International Edition, 2017, 56, 49, 15612–15616.
DOI: 10.1002/anie.201708790
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Development and evaluation of β-galactosidase-sensitive antibody-drug conjugates
Sergii Kolodych, Chloé Michel, Sébastien Delacroix, Oleksandr Koniev, Anthony Ehkirch, Jitka Eberova, Sarah Cianférani, Brigitte Renoux, Wojciech Krezel, Pauline Poinot, Christian D. Muller, Sébastien Papot, Alain Wagner, European Journal of Medicinal Chemistry, 2017, 142, 376-382.

DOI: 10.1016/j.ejmech.2017.08.008
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An in vivo strategy to counteract post-administration anticoagulant activity of azido-Warfarin 
Sylvain Ursuegui,  Marion Recher,  Wojciech Krężel, Alain Wagner. Nature Comm., 2017, 8, 15242.
DOI: 10.1038/ncomms15242

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Acyl Fluorides: Fast, Efficient, and Versatile Lysine-Based Protein Conjugation via Plug-and-Play Strategy.
Igor
Dovgan, Sylvain Ursuegui, Stéphane Erb, Chloé Michel, Sergii Kolodych, Sarah Cianférani, Alain Wagner.  Bioconjugate Chem., 2017, 28, 5, 1452-1457.
DOI: 10.1021/acs.bioconjchem.7b00141

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2016


pH-Responsive Nanometric Polydiacetylenic Micelles Allow for Efficient Intracellular siRNA Delivery.
Manon Ripoll, Patrick Neuberg, Antoine Kichler, Nassera Tounsi, Alain Wagner, Jean-Serge Remy. ACS Appl Mater Interfaces, 2016, 8, 45, 30665–30670.
DOI: 10.1021/acsami.6b09365

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​Copper-free click chemistry for microdroplet's W/O interface engineering.
Sylvain Ursuegui, Michel Mosser, Alain Wagner. RSC Advances, 2016, 6, 97, 94942 – 94948.
DOI: 10.1039/C6RA20385J

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​Ultrafast Click Chemistry with Fluorosydnones.
Hui Liu, Davide Audisio, Lucie Plougastel, Elodie Decuypere, David-Alexandre Buisson, Oleksandr Koniev, Sergii Kolodych, Alain Wagner, Mourad Elhabiri, Anna Krzyczmonik, Sarita Forsback, Olof Solin, Véronique Gouverneur, Frédéric Taran. 
Angewandte Chemie Int. Ed., 2016, 55, 39, 12073 –12077.
Doi: 10.1002/anie.201606495
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​2-(Maleimidomethyl)-1,3-Dioxanes (MD): a Serum-Stable Self-hydrolysable Hydrophilic Alternative to Classical Maleimide Conjugation.
Igor Dovgan, Sergii Kolodych, Oleksandr Koniev, Alain Wagner.
 Nature Scientific Report, 2016, 6, 1, 30835-30840.
DOI: 10.1038/srep30835
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Palladium Catalyzed Chemoselective and Biocompatible Functionalization of Cysteine-Containing Molecules at Room Temperature.
Riyadh Ahmed Atto Al-Shuaeeb, Sergii Kolodych, Oleksandr Koniev, Sébastien Delacroix, Stéphane Erb, Stéphanie Nicolaÿ, Jean-Christophe Cintrat, Jean-Daniel Brion, Sarah Cianférani, Mouâd Alami, Alain Wagner, Samir Messaoudi. Chem. Eur. J., 2016, 22, 32, 11365 – 11370.
DOI: 10.1002/chem.201602277

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​From solution to in-cell study of the chemical reactivity of acid sensitive functional groups: a rational approach towards improved cleavable linkers for biospecific endosomal release. 
Sylvain A. Jacques, Geoffray Leriche, Michel Mosser, Marc Nothisen, Christian D. Muller, Jean-Serge Remy, Alain Wagner. 
Org. Biomol. Chem., 2016, 14, 21, 4794–4803.
DOI: 10.1039/C6OB00846A

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2015


Mannoside Glycolipid Conjugates Display Anti-inflammatory Activity by Inhibition of Toll-like Receptor-4 Mediated Cell Activation.
Vincent Flacher, Patrick Neuberg, Floriane Point, François Daubeuf, Quentin Muller, David Sigwalt, Jean-Daniel Fauny, Jean-Serge Remy, Nelly Frossard, Alain Wagner, Christophe G. Mueller, Evelyne Schaeffer. A
CS Chem. Biol., 2015, 10, 12, 2697–2705.
Doi: 10.1021/acschembio.5b00552

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MAPN: First-in-Class Reagent for kinetically Resolved Thiol-to-Thiol Conjugation
Oleksandr Koniev, Sergii Kolodych, Zoljargal Baatarkhuu, Johann Stojko, Jitka Eberova, Jean-Yves Bonnefoy, Sarah Cianférani, Alain Van Dorsselear,  Alain Wagner. 
Bioconjugate Chem., 2015, 26, 9, 1863–1867.
DOI: 10.1021/acs.bioconjchem.5b00440
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Spiro Di-orthoester (SpiDo), a Human Plasma Stable Acid-Sensitive Cleavable Linker for Lysosomal Release
Geoffray Leriche, Marc Nothisen, Nadège Baumlin, Christian D. Muller, Dominique Bagnard, Jean-Serge Remy, Sylvain A. Jacques, A. Wagner, 
Bioconjugate Chem., 2015, 26, 8, 1461-1465.
DOI: 10.1021/acs.bioconjchem.5b00280

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Photopolymerized micelles of diacetylene amphiphile: physical characterization and cell delivery properties
Patrick Neuberg, Aurélia Périno, Emmanuelle Morin-Picardat, Nicolas Anton, Zeinab Darwich, Denis Weltin, Yves Mely, Andrey S. Klymchenko, Jean-Serge Remy, Alain Wagner.
Chem. Commun., 2015, 51, 58, 11595-11598.
DOI: 10.1039/c5cc03820k

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Developments and recent advancements in the field of endogenous amino acid selective bond forming reactions for bioconjugation
Oleksandr Koniev, Alain Wagner. Chem. Soc. Rev., 2015, 44, 5495-5551.
Doi: 10.1039/C5CS00048C
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​Discovery of potent inhibitors of Schistosoma mansoni NAD+ catabolizing enzyme
Sylvain A. Jacques, Isabelle Kuhn, Oleksandr Koniev, Francis Schuber, Frances E. Lund, Alain Wagner, Hélène Muller-Steffner, Esther Kellenberger, J. Med. Chem., 2015, 58, 8, 3582–3592.
DOI: 10.1021/acs.jmedchem.5b00203

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CBTF: New Amine-to-Thiol Coupling Reagent for Preparation of Antibody Conjugates with Increased Plasma Stability
Sergii Kolodych, Oleksandr Koniev, Zoljargal Baatarkhuu, Jean-Yves Bonnefoy, François Debaene, Sarah Cianférani, Alain Van Dorsselaer, Alain Wagner. 
Bioconjugate Chem. 2015, 26, 2, 197–200.
Doi: 10.1021/bc500610g

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Development of models for prediction of the antioxidant activity of derivatives of natural compounds
Rok Martinčič, Igor Kuzmanovski, Alain Wagner, Marjana Novic. 
Analytica Chimica Acta. 2015, 868, 23–35.
DOI: 10.1016/j.aca.2015.01.050

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2014

4-Halogeno-Sydnones for Fast Strain Promoted Cycloaddition with Cyclooctynes
Lucie Plougastel, Oleksandr Koniev, Simon Specklin, Elodie Decuypere, Christophe Créminon, David-Alexandre Buisson, Alain Wagner, Sergii Kolodych, Frédéric Taran. Chem. Commun. 2014, 50, 66, 9376-9378.
Doi: 10.1039/c4cc03816a

Bio-specific and bio-orthogonal chemistries to switch-off the quencher of a FRET-based fluorescent probe: application to living-cell biothiol imaging
Coraline Egloff, Denis Weltin, C. Calligaro, Michel Mosser, Marc Nothisen, Jean-Serge. Rémy, Alain Wagner. 
Chem. Commun. 2014, 50, 70, 10049-10051.
Doi: 10.1039/c4cc03548h


Developments in the Field of Bioorthogonal Bond Forming Reactions—Past and Present Trends Mathias King, Alain Wagner. Bioconjugate Chem. 2014, 25, 5, 825–839.
Doi: 10.1021/bc500028d

Copper-Chelating Azides for Efficient Click Conjugation Reactions in Complex Media

Valentina Bevilacqua, Mathias King, Manon Chaumontet, Marc Nothisen, Sandra Gabillet, David Buisson, Céline Puente, Alain Wagner, Frédéric Taran. Angewandte Chemie. 2014, 53 ,23, 5972–5976.
Doi: 10.1002/anie.201310671

Selective Irreversible Chemical Tagging of Cysteine with 3-Arylpropiolonitriles
Oleksandr Koniev, Geoffray Leriche, Marc Nothisen, Jean-Serge Remy, Jean-Marc Strub, Christine Schaeffer-Reiss, Alain Van Dorsselaer, Rachid Baati, Alain Wagner. 
Bioconjugate Chem. 2014, 25, 2, 202–206.
Doi: 10.1021/bc400469d

Probing the catalytic mechanism of bovine CD38/NAD+glycohydrolase by site-directed mutagenesis of key active site residues
Isabelle Kuhn, Esther Kellenberger, Cé, line Cakir-Kiefer, Hélène Muller-Steffner, Francis Schuber. Biochim. 
Biophys Acta. 2014, 1844, 7, 1317-1331​.
Doi: 10.1016/j.bbapap.2014.03.014

2013

​Schistosoma mansoni NAD+ catabolizing enzyme : identification of key residues in catalysis
Isabelle Kuhn, Esther Kellenberger, Francis Schuber,  Hélène Muller-Steffner. 
Biochim. Biophys. Acta. 2013, 1834, 12, 2520-2527.
Doi: 10.1016/j.bbapap.2013.09.002

Dynamic Micelles of Mannoside Glycolipids are more Efficient than Polymers for Inhibiting HIV-1 Trans-infection
Evelyne Schaeffer, Laure Dehuyser, David Sigwalt, Vincent Flacher, Serena Bernacchi, Olivier Chaloin, Jean-Serge Remy, Christophe G. Mueller, Rachid Baati, Alain Wagner, 
Bioconjugate Chem. 2013, 24, 11, 1813-1823.
Doi: 10.1021/bc4000806

A new series of Cs+, K+ and Na+ chelators: synthesis, kinetics, thermodynamics and modeling
Alexandre Korovitch, Antoine Le Roux, Florent Barbault, Miryana Hémadi, Nguyêt-Thanh Ha-Duong, Claude Lion, Alain Wagner, Jean-Michel El Hage Chahine, 
Inorganica Chimica Acta, 2013, 394, 45-57.
Doi:10.1016/J.ICA.2012.08.009

2012

Towards a KCC2 blocker pharmacophore model
Florence Lebon, Cécile Pegurier, Marie Ledecq, Benoit Mathieu, Nathalie Bosman, Anne Frycia, Sébastien Lengelé, Kashinath Dhurke, Ananda Kumar Kanduluru, Stéphane Meunier, Alain Wagner, Christian Wolff, Laurent Provins. 
Bioorganic & Medicinal Chemistry Letters. 2012, 22, 12, 3978-3982.
Doi: 10.1016/j.bmcl.2012.04.097

First steps towards conformationally selective artificial lectins: the chair-boat discrimination by molecularly imprinted polymers
Vincent Lemau de Talancé,  Olivier Massinon, Rachid Baati, Alain Wagner, Stéphane P. Vincent. Chemical Communications.
2012, 48, 86, 10684-10686.
Doi: 10.1039/c2cc35386e
 
New tetramethylthiepinium (TMTI) for copper-free click chemistry
Mathias King, Rachid Baati, Alain Wagner. 
Chemical Communication, 2012, 48, 74, 9308 – 9309.
Doi: 10.1039/C2CC35034C

Synthesis of Novel Mannoside Glycolipid Conjugates for Inhibition of HIV-1 Trans-Infection

Laure Dehuyser, Evelyne Schaeffer, Olivier Chaloin, Christophe G. Mueller, Rachid Baati, Alain Wagner. Bioconjugate Chem. 2012, 23, 9, 1731–1739.
DOI: 10.1021/bc200644d


Capillary electrophoresis–inductively coupled plasma-mass spectrometry hyphenation for the determination at the nanogram scale of metal affinities and binding constants of phosphorylated ligands
Fanny Varenne, Mélanie Bourdillon, Michel Meyer, Yi Lin, Marie Brellier, Rachid Baati, Loïc J. Charbonnière, Alain Wagner, Eric Doris, Frédéric Taran, Agnès Hagège. 
Journal of Chromatography A. 2012, 1229, 280–287
Doi: 10.1016/j.chroma.2012.01.066

​A FRET-based probe with a chemically deactivatable quencher
Geoffray Leriche, Ghyslain Budin,  Zeinab Darwich, Denis Weltin, Yves Mély, Andrey S. Klymchenko, Alain Wagner. Chemical Communication 
2012, 48, 26, 3224-3226.
DOI: 10.1039/c2cc17542h

Insights into the mechanism of bovine CD38/NAD+glycohydrolase from the X-Ray structures of its Michaelis Complex and covalently-trapped intermediates

Pascal F. Egea, Hélène Muller-Steffner, Isabelle Kuhn, Céline Cakir-Kiefer, Norman J. Oppenheimer, Robert M. Stroud, Esther Kellenberger, Francis Schuber. 
PLOS One. 2012, 7, 4, 34918.
Doi: 10.1371/journal.pone.0034918

 
Mild chemo-selective hydration of terminal alkynes catalyzed by AgSbF6
Mathieu Bui The Thuong, André Mann, Alain Wagner. Chemical Communication, 2012, 48, 3, 434-436.
Doi: 10.1039/c1cc12928g

Trimethoxyarene, a Highly Ionisable Tag for Reaction Analysis by APPI/MS: Exploration of Heterocyclic Synthesis
Mathieu Bui The Thuong, Cédric Catala,  Cyril Colas, Christine Schaeffer, Alain Van Dorsselaer, André Mann, Alain Wagner. European Journal of Organic Chemistry, 
2012, 2012, 1, 85-92.
Doi: 10.1002/ejoc.201100919

Cleavable linkers in chemical biology
Geoffray Leriche, Louise Chisholm, Alain Wagner. Bioorganic and Medicinal Chemistry. 2012,
 20, 2, 571-582.
Doi: 10.1016/j.bmc.2011.07.048

2011

Flavonoids as inhibitors of human CD38
Esther Kellenberger, Isabelle Kuhn, Francis Schuber, Hélène Muller-Steffner. 
Bioorg Med Chem Lett. 2011, 21, 13, 3939-3942.
Doi: 10.1016/j.bmcl.2011.05.022

Cationic Polydiacetylene Micelles for Gene Delivery
Emmanuelle Morin, Marc Nothisen, Alain Wagner, Jean-Serge Remy. 
Bioconjugate 2011, 22, 10, 1916–1923.
Doi: 10.1021/bc200083p


Self-Assembled Nanotubes and Helical Tapes from Diacetylene Nonionic Amphiphiles. Structural Studies before and after Polymerization
Aurélia Perino, Marc Schmutz, Stéphane Meunier, Philippe J. Mésini, Alain Wagner. 
Langmuir. 2011, 27, 19, 12149–12155.
Doi: 10.1021/la202162q

Structure/function studies of DNA gyrase supramolecular complexes
J. Papillon,  N. Potier,  C. Crucifix, J. F. Menetret, C. Genet, P. Oudet, A.  Wagner, P. Schultz, V. Lamour. 
FEBS Journal. 2011, 278, 472.

Design and synthesis of new antioxidants predicted by the model developed on a set of pulvinic acid derivatives
Antoire Le Roux, Igor Kuzmanovski, Damien Habrant, Stépahne Meunier, Pierre Bischoff, Brice Nadal, Sophie A.-L. Thetiot-Laurent, Thierry Le Gall, Alain Wagner, Marjana Novic. 
Journal of Chemical Information and Modeling. 2011, 51, 12, 3050–3059.
Doi: 10.1021/ci200205d

Stereoselective Addition of Grignard Reagents to New P-Chirogenic N-Phosphinoylbenzaldimines: Effect of the Phosphorus Substituents on the Stereoselectivity
Irene Notar Francesco, Coraline Egloff,  Alain Wagner, Françoise Colobert. 
European Journal of Organic Chemistry. 2011, 20-21, 4037-4045.
Doi: 10.1002/ejoc.201100380

Design, synthesis and evaluation of new α-nucleophiles for the hydrolysis of organophosphorus nerve agents: application to the reactivation of phosphorylated acetylcholinesterase
Géraldine Saint-André, Maria Kliachyna, Sanjeevarao Kodepelly, Ludivine Louise-Leriche, Emilie Gillon, Pierre-Yves Renard, Florian Nachon, Rachid Baati, Alain Wagner. 
Tetrahedron 2011, 67, 34, 6352-6361.
Doi: 10.1016/j.tet.2011.05.130


A Representation to Apply Usual Data Mining Techniques to Chemical Reactions— Illustration on the Rate Constant Of SN2 Reactions in Water
Franck Hoonakker, Nicolas Lachiche, Alexandre Varnek, Alain Wagner. 
International Journal on Artificial Intelligence Tools, 2011, 20, 02, 253-270.
Doi:10.1142/S0218213011000140

First efficient uncharged reactivators for the dephosphylation of poisoned human acetylcholinesterase
Guillaume Mercey, Tristan Verdelet, Géraldine Saint-André, Emilie Gillon, Alain Wagner, Rachid Baati, Ludovic Jean, Florian Nachon, Pierre-Yves Renard. 
Chemical Communication. 2011, 47, 18, 5295-5297.
Doi: 10.1039/c1cc10787a


Programmed Dispersions of MWNTs in Aqueous Media by Coating with Photopolymerizable Synthetic Amphiphiles
Cédric Thauvin, Aurélia Perino, Emmanuel Contal, Emmanuelle Morin, Patrick Schultz, Stéphane Meunier, Alain Wagner. J. Phys. Chem. C. 2011, 115, 15, 7319–7322.
Doi: 10.1021/jp2000464

Synthesis and radioprotective properties of pulvinic acid derivatives
Antoine Le Roux, Stéphane Meunier, Thierry Le Gall, Jean-Marc Denis, Pierre Bischoff, Alain Wagner. 
ChemMedChem. 2011, 6, 3, 561-569.
Doi: 10.1002/cmdc.201000391

Cationic Cyclization of 2-Alkenyl-1,3-dithiolanes: Diastereoselective Synthesis of trans-Decalins

Sylvie Goncalves, Stefano Santoro, Marc Nicolas, Alain Wagner, Philippe Maillos, Fahmi Himo, Rachid Baati. 
Journal of Organic Chemistry. 2011, 76, 9, 3274-3285.
Doi: 10.1021/jo2001116
 

Core functionalization of polydiacetylene micelles by "click" reaction
Emmanuel Contal, Andrey S. Klymchenko, Yves Mély, Stéphane Meunier, Alain Wagner. 
Soft Matter, 2011, 7, 5, 1648-1650.
Doi: 10.1039/C0SM00943A

 
Tailoring drug release profile of low-molecular-weight hydrogels by supramolecular co-assembly and thiol-ene orthogonal coupling
David Díaz Díaz, Emmanuelle Morin, Eva M. Schön, Ghyslain Budin, Alain Wagner, Jean-Serge Remy. 
Journal of Materials Chemistry. 2011, 21, 641-644.
Doi: 10.1039/C0JM03399E


Structure and behaviour of polydiacetylene-based micelles
Aurélia Perino, Andrey S. Klymchenko, Alexandre Morere, Emmanuel Contal, Alain Rameau, Jean-Michel Guenet, Yves Mély, Alain Wagner. Macromolecular Chemistry and Physics. 2011, 212, 2, 111-117.
Doi: 10.1002/macp.201000459

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